This article is cited in 6 papers

First example of cine-substitution for halogens in azolopyrimidines

G. L. Rusinov, P. V. Plekhanov, A. Yu. Ponomareva, O. N. Chupakhin

I. Ya. Postovsky Institute of Organic Synthesis, Urals Branch of the Russian Academy of Sciences, Ekaterinburg, Russian Federation

Abstract: 6-Bromo-1,2,4-triazolo[1,5-a]pyrimidine reacts with indoles in the presence of BF₃ to form σ^H-adducts, which undergo aromatization on treatment with triethylamine.

Language: English

DOI: 10.1070/MC1999v009n06ABEH001126

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